SCHEMBL28655779

SCHEMBL28655779

COC(=O)C1=NN=C2CCN(C(=O)OC(C)(C)C)C=C21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.38
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
GPR119 Q8TDV5 5/20 0.33
EED O75530 1/20 0.32
RBBP4 Q09028 1/20 0.32
SUZ12 Q15022 1/20 0.32
EZH2 Q15910 1/20 0.32
AEBP2 Q6ZN18 1/20 0.32
ALDH1A1 P00352 2/20 0.32
UCHL1 P09936 1/20 0.32
USP30 Q70CQ3 1/20 0.32
ESR2 Q92731 1/20 0.32
GRM5 P41594 1/20 0.31
SETD7 Q8WTS6 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
PTPN2 P17706 1/20 0.31
PTPN1 P18031 1/20 0.31
PTPN6 P29350 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587841 0.86 ADORA1 (0.38) GPR119ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL28696148 0.74 NR1H2 (0.38) NR1H2HDAC1HDAC6GPR119EED
SCHEMBL28449477 0.70 USP2 (0.36) NR1H2GPR119ALDH1A1ESR2GRM5
SCHEMBL20690515 0.70 ALDH1A1 (0.40) NR1H2GPR119ALDH1A1ESR2LMNA
SCHEMBL2980997 0.68 ESR2 (0.43) NR1H2GPR119ALDH1A1ESR2LMNA
SCHEMBL17481737 0.68 USP2 (0.41) NR1H2GPR119ALDH1A1ESR2LMNA
SCHEMBL28686795 0.68 ESR2 (0.34) NR1H2GPR119ESR2GRM5USP2
SCHEMBL29100795 0.68 ESR2 (0.34) NR1H2GPR119ESR2GRM5USP2
SCHEMBL31729924 0.67 CA1 (0.42) NR1H2HDAC1HDAC6ALDH1A1UCHL1
SCHEMBL17942084 0.65 GPR119 (0.39) NR1H2GPR119ALDH1A1ESR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113767101-A Novel indole-2-carboxamides having anti-Hepatitis B Virus (HBV) activity 艾库里斯有限及两合公司 2021-12-07 CN disclosed