SCHEMBL28657384

SCHEMBL28657384

OC1(c2ccccc2)CC(COCc2ccccc2)C1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSK P43235 1/20 0.43
TACR1 P25103 1/20 0.41
OPRL1 P41146 1/20 0.41
NAAA Q02083 1/20 0.40
AGTR2 P50052 1/20 0.40
POLB P06746 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
LMNA P02545 1/20 0.39
BUB1 O43683 1/20 0.39
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9394261 0.85 TSHR (0.48) TSHRCTSLCTSBCTSKNAAA
SCHEMBL5787333 0.83 OPRL1 (0.49) OPRL1POLB
SCHEMBL599216 0.82 TSHR (0.45) TSHRCTSLCTSBCTSKNAAA
SCHEMBL31034964 0.80 TRPV6 (0.42) TSHRCTSLCTSBCTSKTAAR1
SCHEMBL1613917 0.78 TSHR (0.48) TSHRCTSLCTSBCTSKNAAA
SCHEMBL7936478 0.77 AGTR2 (0.45) TSHRCTSLCTSBCTSKNAAA
SCHEMBL20284995 0.77 OPRL1 (0.51) CTSLCTSBCTSKTACR1OPRL1
SCHEMBL20455696 0.76 OPRM1 (0.42) CTSLCTSBCTSKOPRL1
SCHEMBL25631052 0.75 TAAR1 (0.47) TSHRCTSLCTSBCTSKNAAA
SCHEMBL5790770 0.75 CTSL (0.48) TSHRCTSLCTSBCTSKNAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113636977-B Synthesis method of 2-aryl benzazepine and derivatives thereof 温州大学 2022-12-20 CN disclosed
CN-113636977-A Synthesis method of 2-aryl benzazepine and derivatives thereof 温州大学 2021-11-12 CN disclosed