SCHEMBL28658592

SCHEMBL28658592

FC(F)(F)Oc1c[nH]c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 2/20 0.50
GPR84 Q9NQS5 2/20 0.46
MAPK1 P28482 1/20 0.46
STING1 Q86WV6 1/20 0.46
KIF11 P52732 1/20 0.45
ATM Q13315 1/20 0.44
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
AHR P35869 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
PBRM1 Q86U86 1/20 0.42
NR4A2 P43354 1/20 0.41
GOT1 P17174 1/20 0.40
IMPDH2 P12268 1/20 0.40
IMPDH1 P20839 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27704617 0.81 GPR84 (0.53) GPR84MAPK1STING1KIF11CYP3A4
SCHEMBL21965348 0.81 SLC22A6 (0.54) SLC22A6GPR84KIF11ATMMEN1
SCHEMBL28961088 0.78 SLC22A6 (0.55) SLC22A6GPR84MAPK1ATMMEN1
SCHEMBL7086161 0.77 GPR84 (0.62) GPR84MEN1CYP3A4MAPTAHR
SCHEMBL3538344 0.77 SLC22A6 (0.58) SLC22A6GPR84ATMMEN1CYP3A4
SCHEMBL6535531 0.77 SLC22A6 (0.58) SLC22A6GPR84ATMMEN1CYP3A4
SCHEMBL29761872 0.76 TRPA1 (0.51) MAPK1MEN1CYP3A4MAPTAHR
SCHEMBL12475825 0.76 TRPA1 (0.51) MAPK1MEN1CYP3A4MAPTAHR
SCHEMBL10920865 0.75 SLC22A6 (0.53) SLC22A6GPR84MAPK1ATMMEN1
SCHEMBL3925907 0.74 SLC22A6 (0.64) SLC22A6GPR84MAPK1STING1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113717090-B Trifluoromethyl-containing all-carbon quaternary carbon center indole acetonitrile compound and preparation method and application thereof 南京林业大学 2022-04-05 CN disclosed
CN-113717090-B Trifluoromethyl-containing all-carbon quaternary carbon center indole acetonitrile compound and preparation method and application thereof 南京林业大学 2022-04-05 CN disclosed
CN-113717090-A Trifluoromethyl-containing all-carbon quaternary carbon center indole acetonitrile compound and preparation method and application thereof 南京林业大学 2021-11-30 CN disclosed
CN-113717090-A Trifluoromethyl-containing all-carbon quaternary carbon center indole acetonitrile compound and preparation method and application thereof 南京林业大学 2021-11-30 CN disclosed