SCHEMBL28677805

SCHEMBL28677805

O=C(Nc1cccc2ccccc12)c1cccnc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.78
CYP1A2 P05177 2/20 0.78
CYP2C19 P33261 2/20 0.78
KDM4E B2RXH2 2/20 0.78
L3MBTL1 Q9Y468 2/20 0.71
CYP2C9 P11712 2/20 0.69
NPC1 O15118 2/20 0.69
RAB9A P51151 2/20 0.69
CYP3A4 P08684 1/20 0.69
CYP2D6 P10635 1/20 0.69
HTT P42858 2/20 0.68
BLM P54132 1/20 0.65
HDAC3 O15379 1/20 0.65
HDAC1 Q13547 1/20 0.65
HDAC2 Q92769 1/20 0.65
SMN1; SMN2 Q16637 3/20 0.64
ALOX15 P16050 1/20 0.62
MAPT P10636 1/20 0.60
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657603 0.88 ALDH1A1 (0.70) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1
SCHEMBL23332048 0.84 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1
SCHEMBL11616061 0.83 RAB9A (0.76) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1
SCHEMBL30184438 0.82 NPC1 (1.00) CYP1A2CYP2C19KDM4ECYP2C9NPC1
SCHEMBL4642544 0.82 NPC1 (1.00) CYP1A2CYP2C19KDM4ECYP2C9NPC1
SCHEMBL17737359 0.82 KMT2A (0.76) ALDH1A1CYP1A2CYP2C19KDM4ECYP2C9
SCHEMBL6645868 0.81 HTT (1.00) ALDH1A1KDM4EL3MBTL1NPC1RAB9A
SCHEMBL4531531 0.81 L3MBTL1 (0.64) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1
SCHEMBL13966176 0.81 L3MBTL1 (0.64) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1
SCHEMBL20421676 0.80 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368083-B Heteroaryl compounds and their use as therapeutic agents 东亚首希控股股份有限公司 2022-02-01 CN disclosed