SCHEMBL28698319

SCHEMBL28698319

Cc1ccc(S(=O)(=O)C2CNCCN2C(C)c2ccc(Br)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.40
CHRM1 P11229 2/20 0.40
CCR5 P51681 1/20 0.34
MAPT P10636 2/20 0.34
RECQL P46063 2/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
HTT P42858 1/20 0.34
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HTR2C P28335 1/20 0.33
HTR6 P50406 1/20 0.33
HSD11B1 P28845 8/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27845743 0.74 CHRM2 (0.38) CHRM2CHRM1LMNAGAAHTR2C
SCHEMBL4839034 0.74 CCR5 (0.44) CHRM2CHRM1CCR5HTR2CHSD11B1
SCHEMBL10073178 0.72 ADRB1 (0.41) CHRM2CHRM1CCR5HTR2CHTR6
SCHEMBL11628818 0.72 L3MBTL1 (0.47) MAPTRECQLHTTLMNAHTR2C
SCHEMBL9120393 0.71 ADRB1 (0.38) CHRM2CHRM1MAPTRECQLHTT
SCHEMBL30754657 0.70 ALDH1A1 (0.40) HPGDHTR2CHTR6ALDH1A1
SCHEMBL3822494 0.69 CACNA2D1 (0.41) CHRM2CHRM1ATMALDH1A1
SCHEMBL23646035 0.68 ALDH1A1 (0.37) HTTHTR2CHTR6ALDH1A1
SCHEMBL736080 0.68 CA1 (0.50) MAPTHPGDLMNAGAAALDH1A1
SCHEMBL2266732 0.68 LMNA (0.65) CHRM2CHRM1HTTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115776983-A Heterocyclic immunomodulators 北京诺诚健华医药科技有限公司 2023-03-10 CN disclosed
CN-113896711-A Heterocyclic immunomodulators 北京诺诚健华医药科技有限公司 2022-01-07 CN disclosed