SCHEMBL28706015

SCHEMBL28706015

O=C(O)N1CC2N(Cc3ccccc3)C(=O)C(O)C2(F)C1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
EHMT2 Q96KQ7 1/20 0.38
BRD4 O60885 1/20 0.36
HSD11B1 P28845 1/20 0.35
FUCA1 P04066 2/20 0.35
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
RIPK1 Q13546 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29471673 0.85 RORC (0.41) SMN1; SMN2GAA
SCHEMBL16714596 0.69 CYP19A1 (0.44) TSHRCYP3A4CYP2C19MEN1KMT2A
SCHEMBL26965338 0.67 RIPK1 (0.41) TSHRCYP2C19MEN1KMT2AALDH1A1
SCHEMBL28701185 0.67 GRM6 (0.41) TSHRMEN1KMT2AHSD11B1ALDH1A1
SCHEMBL22950454 0.65 RORC (0.42)
SCHEMBL20722495 0.64 S1PR5 (0.49) TSHRMEN1KMT2AHSD11B1FUCA1
SCHEMBL28612669 0.64 AMPD2 (0.37) TSHRCYP3A4MEN1KMT2ABRD4
SCHEMBL21682573 0.64 AMPD2 (0.37) TSHRCYP3A4MEN1KMT2ABRD4
SCHEMBL17685922 0.63 BRD4 (0.52) EHMT2BRD4
SCHEMBL15719254 0.62 CTSL (0.40) CYP2C19ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114173787-A Dihydropyrimidine derivatives and their use in the treatment of HBV infection or HBV-induced diseases 杨森科学爱尔兰无限公司 2022-03-11 CN disclosed