SCHEMBL28708243

SCHEMBL28708243

COc1ccccc1NC(=O)N[C@H]1CCN(C(=O)O)C1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.58
CA12 O43570 2/20 0.56
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA4 P22748 2/20 0.56
CA7 P43166 2/20 0.56
CA9 Q16790 2/20 0.56
ALDH1A1 P00352 4/20 0.54
TAS1R3 Q7RTX0 1/20 0.54
TAS1R1 Q7RTX1 1/20 0.54
ACHE P22303 1/20 0.54
BACE1 P56817 1/20 0.54
SIGMAR1 Q99720 1/20 0.53
TSHR P16473 1/20 0.52
PKM P14618 1/20 0.51
MAPK1 P28482 1/20 0.51
DRD2 P14416 1/20 0.51
ADRA1D P25100 1/20 0.51
ADRA1A P35348 1/20 0.51
ADRA1B P35368 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31616468 0.82 SIGMAR1 (0.71) ALDH1A1SIGMAR1TSHRDRD2KMT2A
SCHEMBL31616372 0.82 SIGMAR1 (0.71) ALDH1A1SIGMAR1TSHRDRD2KMT2A
SCHEMBL2752062 0.79 TAS1R3 (0.71) POLBALDH1A1TAS1R3TAS1R1TSHR
SCHEMBL20365400 0.78 KMT2A (0.72) POLBALDH1A1TAS1R3TAS1R1MAPK1
SCHEMBL6684742 0.78 BRD4 (0.64) ALDH1A1ACHEBACE1PKMMAPK1
SCHEMBL6663459 0.77 CHRM3 (0.58) ACHEBACE1KMT2AL3MBTL1
SCHEMBL6667431 0.77 ACHE (0.57) POLBALDH1A1ACHEBACE1TSHR
SCHEMBL5458362 0.76 RAB9A (0.58) CA12CA1CA2CA9ALDH1A1
SCHEMBL10542205 0.76 POLB (0.60) POLBALDH1A1TAS1R3TAS1R1PKM
SCHEMBL1911204 0.75 RECQL (0.54) POLBCA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed