SCHEMBL28709587

SCHEMBL28709587

O=C(c1cc(-c2ccccc2)ccc1[N+](=O)[O-])N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
BLM P54132 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
HTT P42858 2/20 0.52
LMNA P02545 1/20 0.52
FAAH O00519 2/20 0.51
PRKAB2 O43741 2/20 0.50
PRKAG1 P54619 2/20 0.50
PRKAA2 P54646 2/20 0.50
PRKAA1 Q13131 2/20 0.50
PRKAG3 Q9UGI9 2/20 0.50
PRKAG2 Q9UGJ0 2/20 0.50
PRKAB1 Q9Y478 2/20 0.50
MGLL Q99685 1/20 0.49
MAPK1 P28482 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28706683 0.91 FAAH (0.54) SIGMAR1BLML3MBTL1HTTLMNA
SCHEMBL28715872 0.88 BLM (0.50) BLML3MBTL1HTTLMNAFAAH
SCHEMBL28716592 0.83 ALDH1A1 (0.53) BLML3MBTL1HTTLMNAFAAH
SCHEMBL30525110 0.82 SIGMAR1 (0.49) SIGMAR1L3MBTL1LMNAFAAHPRKAB2
SCHEMBL30525111 0.74 FAAH (0.48) SIGMAR1HTTLMNAFAAHALDH1A1
SCHEMBL30064690 0.74 SIGMAR1 (0.66) SIGMAR1L3MBTL1FAAHPRKAB2PRKAG1
SCHEMBL27629355 0.71 SIGMAR1 (0.68) SIGMAR1L3MBTL1FAAHPRKAB2PRKAG1
SCHEMBL6706057 0.71 MCHR1 (0.59) ALDH1A1MAPT
SCHEMBL15687847 0.70 HPD (0.52) LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL15842125 0.70 RORC (0.71) SIGMAR1L3MBTL1LMNAPRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461640-A LPAR1 inhibitor, medical application and preparation method thereof 中央民族大学 2021-10-01 CN claimed
CN-113461640-A LPAR1 inhibitor, medical application and preparation method thereof 中央民族大学 2021-10-01 CN disclosed