SCHEMBL287419

SCHEMBL287419

O=C(CN(Nc1ccccn1)C(=O)C1=CN=CCC1)c1cccs1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.41
RAB9A P51151 7/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CTNNB1 P35222 1/20 0.40
SMN1; SMN2 Q16637 7/20 0.39
GAA P10253 1/20 0.39
ESR1 P03372 1/20 0.36
POLB P06746 1/20 0.36
STAT3 P40763 1/20 0.36
ESR2 Q92731 1/20 0.36
PKM P14618 2/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
OPRM1 P35372 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287307 0.84 ALDH1A1 (0.39) NPC1RAB9AKMT2ASMN1; SMN2POLB
SCHEMBL287408 0.80 RAB9A (0.43) NPC1RAB9AKMT2AHSD17B10SMN1; SMN2
SCHEMBL287518 0.80 ALDH1A1 (0.35) NPC1RAB9AKMT2ASMN1; SMN2ESR1
SCHEMBL287274 0.77 ALDH1A1 (0.33) NPC1RAB9AKMT2ACTNNB1SMN1; SMN2
SCHEMBL287825 0.75 ALDH1A1 (0.34) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1
SCHEMBL287139 0.74 ALDH1A1 (0.38) NPC1RAB9AKMT2AHSD17B10CTNNB1
SCHEMBL286788 0.73 MAPT (0.35) NPC1RAB9AKMT2AHSD17B10SMN1; SMN2
SCHEMBL288004 0.73 ALDH1A1 (0.48) NPC1RAB9AKMT2ASMN1; SMN2GAA
SCHEMBL287767 0.73 HPGD (0.42) NPC1RAB9AKMT2APOLBALDH1A1
SCHEMBL287813 0.72 ALDH1A1 (0.45) NPC1RAB9AKMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP claimed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO claimed