SCHEMBL28746461

SCHEMBL28746461

CCOC(=O)c1c(C)nc(-c2ccccc2Cl)n1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.53
PDE2A O00408 1/20 0.52
PDE10A Q9Y233 1/20 0.52
MAPT P10636 4/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
TP53 P04637 2/20 0.49
RAB9A P51151 2/20 0.49
HCRTR1 O43613 1/20 0.49
ALOX15 P16050 1/20 0.49
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 3/20 0.47
HPGD P15428 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PDE4B Q07343 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LMNA P02545 2/20 0.46
CDC7 O00311 1/20 0.46
DBF4 Q9UBU7 1/20 0.46
GRM6 O15303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746444 0.88 F11 (0.48) MAPK1PDE2APDE10AMAPTSMN1; SMN2
SCHEMBL29565489 0.88 F11 (0.48) MAPK1PDE2APDE10AMAPTSMN1; SMN2
SCHEMBL28746453 0.82 LMNA (0.51) MAPK1SMN1; SMN2RAB9AALDH1A1KDM4E
SCHEMBL25326523 0.81 KDM4E (0.47) MAPK1MAPTSMN1; SMN2TP53RAB9A
SCHEMBL25328154 0.81 CYP1A2 (0.66) MAPK1MAPTSMN1; SMN2TP53RAB9A
SCHEMBL28746434 0.78 MAPT (0.56) MAPTSMN1; SMN2TP53RAB9AALDH1A1
SCHEMBL29565728 0.77 TRPM8 (0.53) MAPK1MAPTSMN1; SMN2TP53RAB9A
SCHEMBL28746466 0.77 TRPM8 (0.53) MAPK1MAPTSMN1; SMN2TP53RAB9A
SCHEMBL28746474 0.75 MAPK1 (0.43) MAPK1PDE2APDE10AMAPTSMN1; SMN2
SCHEMBL28800164 0.74 PDE4B (0.55) MAPK1PDE2APDE10AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539158-B FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2023-12-08 CN disclosed
CN-114539158-A FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2022-05-27 CN disclosed