SCHEMBL28760040

SCHEMBL28760040

CCC(C)C(=N)c1nc(-c2ccc(F)c(Cl)c2)cc(N2CCNCC2)n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 4/20 0.41
JAK2 O60674 1/20 0.39
SOS1 Q07889 5/20 0.36
PRKD1 Q15139 2/20 0.36
PRKD2 Q9BZL6 2/20 0.36
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
P2RY12 Q9H244 1/20 0.36
PTPN11 Q06124 2/20 0.35
INPPL1 O15357 1/20 0.35
KMO O15229 1/20 0.35
TRPV3 Q8NET8 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27656893 0.84 TRPV3 (0.35) ALKPTPN11KMOTRPV3
SCHEMBL27635865 0.80 TRPV1 (0.35) HRH4PTPN11KMOTRPV3
SCHEMBL907895 0.73 CETP (0.42) SOS1HRH4HRH3PTPN11
SCHEMBL908061 0.70 CASP1 (0.39) SOS1PRKD1PRKD2HRH4HRH3
SCHEMBL27635880 0.69 KIT (0.34)
SCHEMBL27635905 0.68 ADORA3 (0.36) TRPV3
SCHEMBL3881055 0.64 EPHX2 (0.54)
SCHEMBL27635986 0.62 HSD11B1 (0.44)
SCHEMBL3876842 0.61 HSD11B1 (0.49)
SCHEMBL25409176 0.61 SOS1 (0.39) SOS1PTPN11HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1823057-A Biaryl piperazinyl-pyridine analogues NEUROGEN CORP (US) 2006-08-23 CN disclosed