SCHEMBL28778792

SCHEMBL28778792

CC1(C)CNCCN1c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LIPE Q05469 3/20 0.40
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
SCN4A P35499 1/20 0.36
SCN9A Q15858 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CCR6 P51684 4/20 0.36
KCNH2 Q12809 3/20 0.36
NISCH Q9Y2I1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27728779 0.99 SLC6A4 (0.45) SLC6A4SLC6A2SLC6A3POLBL3MBTL1
SCHEMBL28780742 0.85 PIM1 (0.43) SLC6A4SLC6A2SLC6A3ADRB1KCNH2
SCHEMBL3017728 0.82 ADRB1 (0.56) POLBALDH1A1HTR3EHTR3BADRB1
Hydrochloric Acid SCHEMBL2524208 0.81 ADRB1 (0.54) POLBALDH1A1HTR3EHTR3BADRB1
SCHEMBL27728780 0.77 ALDH1A1 (0.50) SLC6A4SLC6A2SLC6A3ALDH1A1TSHR
SCHEMBL7647236 0.77 ADRB1 (0.52) POLBALDH1A1ADRB1HTR2AHTR2C
SCHEMBL27744781 0.77 SLC6A4 (0.43) SLC6A4SLC6A2SLC6A3LIPEALDH1A1
SCHEMBL19003593 0.76 MGLL (0.39) POLBL3MBTL1ALDH1A1ADRB1KCNH2
SCHEMBL7943366 0.75 MAPT (0.38) POLBL3MBTL1ALDH1A1HTR3EHTR3B
SCHEMBL4487460 0.75 ADRB1 (0.50) SLC6A4SLC6A2SLC6A3HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101421258-B Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYPSYS INC 2013-08-21 CN disclosed
CN-101421258-A Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYSPSYS INC (US) 2009-04-29 CN disclosed
CN-101374813-A Arylsulfonamide and sulfonyl compounds as PPAR modulators and methods of treating metabolic disorders KALYPSYS INC (US) 2009-02-25 CN disclosed