SCHEMBL28782010

SCHEMBL28782010

CS(=O)(=O)CCn1cc2ccccc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
KEAP1 Q14145 1/20 0.35
TP53 P04637 1/20 0.34
ALDH1A1 P00352 2/20 0.34
NQO2 P16083 1/20 0.34
HTR6 P50406 1/20 0.33
POLR1A O95602 1/20 0.32
HSD17B10 Q99714 1/20 0.31
USP2 O75604 2/20 0.31
MEN1 O00255 1/20 0.31
ESR1 P03372 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CASP1 P29466 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CNR1 P21554 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28199765 0.72 TP53 (0.65) TP53ALDH1A1
SCHEMBL377726 0.72 CDK4 (0.33) HTTALDH1A1CA12BRD4BRPF1
SCHEMBL16235881 0.69 ALDH1A1 (0.41) HTTTP53ALDH1A1USP2MEN1
SCHEMBL6750562 0.68 HTT (0.37) HTTALDH1A1USP2MEN1ESR1
SCHEMBL5729887 0.68 ALDH1A1 (0.44) TP53ALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL3632871 0.67 BCHE (0.34) ALDH1A1
SCHEMBL7004471 0.67 HTR2A (0.38) ALDH1A1HTR6HSD17B10SMN1; SMN2CA12
SCHEMBL14524221 0.67 KEAP1 (0.36) HTTKEAP1ALDH1A1NQO2HTR6
SCHEMBL1306411 0.67 GLS (0.53) MEN1CYP1A2CYP2C19KMT2ACA9
SCHEMBL10412639 0.66 CYP2A6 (0.37) HTTTP53ALDH1A1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511840-A Phosphoinositide 3-kinase inhibitor compounds and methods of use thereof GENENTECH INC (US) 2009-08-19 CN disclosed