SCHEMBL28787697

SCHEMBL28787697

CC(=O)Oc1coc(-c2cccc(Cl)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
IKBKB O14920 1/20 0.44
NPC1 O15118 5/20 0.43
RAB9A P51151 4/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NOTUM Q6P988 3/20 0.42
PTGS2 P35354 1/20 0.41
KMT2A Q03164 2/20 0.41
PDE4B Q07343 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
TSHR P16473 3/20 0.40
ADORA2A P29274 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
MAPT P10636 2/20 0.40
ABL1 P00519 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27539135 0.84 LMNA (0.40) NPC1RAB9AL3MBTL1PDE4BSMN1; SMN2
SCHEMBL27516569 0.83 LMNA (0.53) NPC1RAB9AL3MBTL1TSHRADORA2A
SCHEMBL17360640 0.80 HDAC1 (0.54) NPC1RAB9ANOTUMKMT2ASMN1; SMN2
SCHEMBL28742829 0.78 HPGD (0.41) FFAR1NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL4640428 0.76 MAPK1 (0.47) NPC1RAB9AL3MBTL1KMT2ASMN1; SMN2
SCHEMBL1544536 0.76 HDAC1 (0.50) FFAR1IKBKBNOTUMPDE4BTP53
SCHEMBL2868465 0.74 ADRB2 (0.55) FFAR1IKBKBNPC1RAB9AL3MBTL1
SCHEMBL27515881 0.74 NPC1 (0.39) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL27539429 0.74 MAPT (0.35) NPC1RAB9AL3MBTL1PTGS2KMT2A
SCHEMBL28815027 0.74 HDAC1 (0.37) NPC1RAB9APDE4BSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101723941-A “1,2,4” oxadiazole as a metabotropic glutamate receptor-5 modulator ASTRAZENECA AB 2010-06-09 CN disclosed