SCHEMBL28790701

SCHEMBL28790701

Cc1ccc(F)cc1NC(=O)Nc1cccc2c1ccn2Cc1c[nH]c2ncccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
HTR2A P28223 3/20 0.42
HTR7 P34969 3/20 0.42
TP53 P04637 2/20 0.39
PDPK1 O15530 1/20 0.38
MTNR1A P48039 1/20 0.38
GAA P10253 1/20 0.37
DRD4 P21917 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
LMNA P02545 2/20 0.37
BRAF P15056 1/20 0.37
ESR1 P03372 1/20 0.37
PTGER3 P43115 2/20 0.37
HTT P42858 2/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27807485 0.90 TRPV1 (0.48) HTR1AHTR2AHTR7TP53PDPK1
SCHEMBL27807477 0.90 DRD4 (0.41) PDPK1MTNR1ADRD4KDM4EALDH1A1
SCHEMBL3699011 0.89 ALDH1A1 (0.45) MTNR1ADRD4KDM4EALDH1A1HPGD
SCHEMBL3711712 0.89 HTR1A (0.44) HTR1AHTR2AHTR7TP53DRD4
Hydrochloric Acid SCHEMBL3706766 0.89 ALDH1A1 (0.44) TP53MTNR1ADRD4KDM4EALDH1A1
SCHEMBL28790687 0.88 TP53 (0.37) TP53GAALMNABRAFESR1
SCHEMBL3699567 0.88 PTGER3 (0.47) HTR1AHTR2AHTR7PDPK1KDM4E
SCHEMBL3705879 0.88 RAB9A (0.46) HTR1AHTR2AHTR7PDPK1MTNR1A
SCHEMBL3704922 0.88 HTR1A (0.42) HTR1AHTR2AHTR7PDPK1MTNR1A
SCHEMBL28787359 0.88 HTR1A (0.42) HTR1AHTR2AHTR7GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102066372-A 5, 6-membered heteroaryl bicyclic compounds containing a urea group as kinase inhibitors ASCEPION PHARMACEUTICALS INC 2011-05-18 CN claimed
CN-102066372-B 5, 6-membered heteroaryl bicyclic compounds containing a urea group as kinase inhibitors ASCEPION PHARMACEUTICALS INC 2014-09-17 CN disclosed
CN-102066372-A 5, 6-membered heteroaryl bicyclic compounds containing a urea group as kinase inhibitors ASCEPION PHARMACEUTICALS INC 2011-05-18 CN disclosed