SCHEMBL28802154

SCHEMBL28802154

O=C(O)N1CCC(CNS(=O)(=O)c2ccccc2F)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
PKM P14618 1/20 0.49
DPP4 P27487 1/20 0.47
GBA1 P04062 2/20 0.47
TGFBR1 P36897 1/20 0.46
CNR2 P34972 4/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
NSD2 O96028 1/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 1/20 0.43
MAPK14 Q16539 1/20 0.43
MAPT P10636 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27917806 0.85 ALDH1A1 (0.52) ALDH1A1PKMGBA1TGFBR1ADRA1A
SCHEMBL27917798 0.84 NPY1R (0.57) ALDH1A1PKMTGFBR1CNR2CYP2C9
SCHEMBL27917809 0.83 NPY5R (0.58) ALDH1A1GBA1NSD2MAPTHPGD
SCHEMBL27917924 0.83 ALDH1A1 (0.70) ALDH1A1PKMGBA1TGFBR1HDAC3
SCHEMBL5848417 0.82 MEN1 (0.57) ALDH1A1GBA1CNR2CYP2C9HDAC3
SCHEMBL5849554 0.82 MEN1 (0.57) ALDH1A1GBA1CNR2CYP2C9HDAC3
SCHEMBL27917833 0.82 TGFBR1 (0.54) ALDH1A1PKMTGFBR1ADRA1AADRA1B
SCHEMBL28805529 0.82 CNR1 (0.48) ALDH1A1PKMTGFBR1CNR2ADRA1A
SCHEMBL14834085 0.81 MGLL (0.67) DPP4TGFBR1CNR2CYP2C9
SCHEMBL18446034 0.80 HTR1A (0.54) ALDH1A1PKMGBA1CNR2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103068797-A Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application SANOFI SA 2013-04-24 CN disclosed