SCHEMBL28802500

SCHEMBL28802500

C[C@@H](C(=N)C[C@](C)(CO)C(=O)OC(C)(C)C)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.36
CTSS P25774 1/20 0.36
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GPR88 Q9GZN0 2/20 0.34
AAK1 Q2M2I8 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
GAA P10253 1/20 0.33
GRM7 Q14831 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27885815 1.00 CTSK (0.36) CTSKCTSSMAPTMEN1KMT2A
SCHEMBL16782694 0.70 APP (0.47) CTSKCTSSMAPTMEN1KMT2A
SCHEMBL2289610 0.70 APP (0.47) CTSKCTSSMAPTMEN1KMT2A
SCHEMBL17721325 0.70 RIPK1 (0.42) CTSKCTSSMAPTAAK1CYP2C19
SCHEMBL27713396 0.68 L3MBTL1 (0.38) CTSKCTSS
SCHEMBL17123620 0.67 RIPK1 (0.46) CTSKCTSSMAPT
SCHEMBL28037817 0.66 MMP8 (0.39) CYP2C19HIF1A
SCHEMBL1951664 0.65 CTSK (0.45) CTSKCTSSMAPTMEN1KMT2A
SCHEMBL28388602 0.65 CTSK (0.45) CTSKCTSSMAPTMEN1KMT2A
SCHEMBL1951580 0.65 CTSK (0.45) CTSKCTSSMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189222-B Tri-, tetra-substituted-3-aminopyrrolidine derivative DAIICHI SANKYO CO LTD 2013-01-02 CN disclosed