SCHEMBL28814958

SCHEMBL28814958

FC(F)(F)COc1ccc2[nH]ncc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 1/20 0.48
TRPA1 O75762 7/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
MAOB P27338 2/20 0.46
METAP2 P50579 2/20 0.45
NOS1 P29475 3/20 0.45
ROCK2 O75116 2/20 0.45
ROCK1 Q13464 2/20 0.45
CSNK2A1 P68400 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP17A1 P05093 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25344307 0.88 METAP2 (0.57) MEN1KMT2APOLBTRPA1METAP2
SCHEMBL10598655 0.79 TRPA1 (0.57) MEN1KMT2ATRPA1TRPM8METAP2
SCHEMBL3537344 0.79 RAB9A (0.60) MEN1KMT2ATRPA1MAOBMETAP2
SCHEMBL25921681 0.76 MAOB (0.47) MEN1KMT2APOLBMAOBMETAP2
SCHEMBL5410655 0.76 ROCK2 (0.50) MEN1KMT2AMAOBMETAP2NOS1
SCHEMBL14863544 0.76 NOS1 (0.50) MEN1KMT2APOLBMAOBMETAP2
SCHEMBL5804533 0.76 MAOB (0.47) MEN1KMT2AMAOBMETAP2NOS1
SCHEMBL16023545 0.76 NOS1 (0.50) MEN1KMT2APOLBTRPA1MAOB
SCHEMBL4980408 0.75 MAOB (0.52) MEN1KMT2AMAOBMETAP2NOS1
SCHEMBL5407397 0.75 KCNH2 (0.49) MEN1KMT2ATRPA1MAOBMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105451737-B Medical composition and its use and described pharmaceutical composition are used for the application process practised contraception on demand 拜耳医药股份有限公司 2018-04-10 CN disclosed
CN-104144922-B 2H-indazoles as EP 2 receptor antagonists 拜耳知识产权有限责任公司 2016-08-31 CN disclosed
CN-105451737-A Pharmaceutical composition and the use thereof, and application regime of said pharmaceutical composition for on-demand contraception Bayer Pharma AG 2016-03-30 CN disclosed
CN-104144922-A As EP2Novel 2H-indazoles as receptor antagonists BAYER IP GMBH 2014-11-12 CN disclosed