SCHEMBL28815005

SCHEMBL28815005

Fc1c(Br)cccc1N=C(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
ESR1 P03372 5/20 0.39
ESR2 Q92731 5/20 0.39
CTSL P07711 2/20 0.36
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
NOS3 P29474 2/20 0.33
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2784971 0.83 GAA (0.46) GAAESR1ESR2NOS3NOS1
SCHEMBL31212333 0.77 ATM (0.43) GAAIDO1TDO2NPC1RAB9A
SCHEMBL25981306 0.77 ATM (0.43) GAAIDO1TDO2NPC1RAB9A
SCHEMBL29220708 0.75 GAA (0.46) GAAESR1ESR2NPC1RAB9A
SCHEMBL14833836 0.74 CTSL (0.47) CTSLNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL14833839 0.74 CTSL (0.47) CTSLNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL25876652 0.72 NOS3 (0.37) GAAESR1ESR2NOS3NOS1
SCHEMBL12479044 0.72 RXRA (0.37) GAAESR1ESR2
SCHEMBL24536162 0.71 GAA (0.38) GAAESR1ESR2
SCHEMBL1494661 0.71 ESR1 (0.39) GAAESR1ESR2CTSLIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114891070-A Anthelmintic depsipeptide compounds 勃林格殷格翰动物保健美国公司 2022-08-12 CN disclosed
CN-107835818-B Anthelmintic depsipeptide compounds 勃林格殷格翰动物保健美国公司 2022-04-29 CN disclosed
CN-107835818-A Anthelmintic depsipeptide compounds 梅里亚股份有限公司 2018-03-23 CN disclosed