SCHEMBL28815568

SCHEMBL28815568

CC(C)(C)OC(=O)N1CCC(c2nnc[nH]2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.56
KDM4E B2RXH2 1/20 0.56
MAPT P10636 1/20 0.56
HPGDS O60760 2/20 0.49
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
TYK2 P29597 1/20 0.48
JAK3 P52333 1/20 0.48
GPR119 Q8TDV5 6/20 0.47
HTT P42858 1/20 0.46
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44
PTPN6 P29350 1/20 0.44
HPGD P15428 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
NAMPT P43490 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18788537 0.93 THRB (0.50) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL4485955 0.83 ALDH1A1 (0.46) THRBKDM4EMAPTHTTGAA
SCHEMBL8550947 0.80 KDM4E (0.51) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL12836454 0.79 JAK3 (0.41) THRBKDM4EMAPTJAK2JAK1
SCHEMBL9965876 0.79 JAK3 (0.41) THRBKDM4EMAPTJAK2JAK1
SCHEMBL948255 0.79 GPR119 (0.53) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL2512441 0.78 KDM4E (0.52) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL459905 0.77 MAPT (0.51) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL2899508 0.77 THRB (0.51) THRBKDM4EMAPTHPGDSJAK2
SCHEMBL16457597 0.77 KDM4E (0.51) THRBKDM4EMAPTHPGDSJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114874186-B Glutamine acyl cyclase isozyme inhibitor and preparation method and application thereof 深圳大学 2023-07-11 CN disclosed
CN-114874186-A Glutaminyl cyclase isoenzyme inhibitor and preparation method and application thereof 深圳大学 2022-08-09 CN disclosed