SCHEMBL28818318

SCHEMBL28818318

Fc1cccc(Cc2cc[c]c(C(F)(F)F)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.40
IDO1 P14902 2/20 0.39
AGXT P21549 2/20 0.39
DAO P14920 2/20 0.38
P2RX7 Q99572 3/20 0.36
MIF P14174 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
IDH1 O75874 1/20 0.35
SLC6A3 Q01959 1/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939775 0.85 CALM1 (0.43) IDH1
SCHEMBL28008868 0.79 CYP17A1 (0.36) DAOALDH1A1
SCHEMBL28009293 0.77 IDO1 (0.39) TAAR1IDO1AGXTDAOMIF
SCHEMBL3300303 0.76 TAAR1 (0.60) TAAR1IDO1AGXTDAOMIF
SCHEMBL27328871 0.75 TAAR1 (0.47) TAAR1IDO1AGXTDAOMIF
SCHEMBL28009286 0.75 PTPN5 (0.37) TAAR1IDO1DAOALDH1A1SMN1; SMN2
SCHEMBL2430768 0.75 NT5E (0.43) TAAR1IDO1
SCHEMBL262756 0.74 NT5E (0.30)
SCHEMBL9900323 0.72
SCHEMBL27944323 0.72 KIF11 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596923-B 1,2, 4-thiazolidin-3-one derivatives and their use in the treatment of cancer BALTIC BIO AB 2015-04-29 CN claimed
CN-102596923-B 1,2, 4-thiazolidin-3-one derivatives and their use in the treatment of cancer BALTIC BIO AB 2015-04-29 CN disclosed