SCHEMBL28819252

SCHEMBL28819252

O=C(C=Cc1ccccc1)C=Cc1ccc(OCC(=O)N2CCN(S(=O)(=O)c3cccs3)CC2)cc1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.76
PKM P14618 10/20 0.76
SMN1; SMN2 Q16637 5/20 0.67
GPR183 P32249 1/20 0.59
LMNA P02545 3/20 0.57
KEAP1 Q14145 1/20 0.53
NFE2L2 Q16236 1/20 0.53
KMT2A Q03164 1/20 0.51
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819249 0.86 ALDH1A1 (0.58) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28948647 0.82 PKM (0.76) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28819229 0.81 PKM (0.59) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28819250 0.80 RAB9A (0.54) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28819246 0.80 ALDH1A1 (0.60) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28819242 0.78 LMNA (0.58) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL28819253 0.77 LMNA (0.79) ALDH1A1PKMSMN1; SMN2GPR183LMNA
SCHEMBL16599355 0.74 GPR183 (1.00) ALDH1A1PKMGPR183KMT2A
SCHEMBL16599356 0.74 GPR183 (1.00) ALDH1A1PKMGPR183KMT2A
SCHEMBL24893097 0.74 MEN1 (0.70) ALDH1A1SMN1; SMN2GPR183LMNAKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634465-B Pentadienone derivative containing sulfonyl piperazine as well as preparation method and application thereof 贵州大学 2023-05-30 CN disclosed
CN-114634465-A Sulfonyl piperazine-containing pentadiene ketone derivative and preparation method and application thereof 贵州大学 2022-06-17 CN disclosed