SCHEMBL28824043

SCHEMBL28824043

O=C(O)c1cnnn1-c1ccc(-c2ccccc2Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
SCN9A Q15858 2/20 0.45
MARS1 P56192 1/20 0.44
EGLN1 Q9GZT9 2/20 0.44
CYP2A6 P11509 1/20 0.42
MAP4K4 O95819 1/20 0.41
HSD11B1 P28845 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
PPP1CA P62136 1/20 0.40
EGLN3 Q9H6Z9 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.39
HSP90AA1 P07900 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949284 0.90 SCN9A (0.45) KMT2AMEN1SCN9AMARS1HSD11B1
SCHEMBL28824045 0.86 RPA1 (0.46) KMT2AMEN1MARS1HSD11B1NPC1
SCHEMBL28823984 0.85 BRS3 (0.43) KMT2ANPC1HSP90AA1NFKB1RAB9A
SCHEMBL28824102 0.84 MAPK9 (0.46) KMT2AMEN1HSD11B1KDM4EALDH1A1
SCHEMBL28824005 0.84 ALDH1A1 (0.42) KMT2AMEN1HSD11B1ALDH1A1NPC1
SCHEMBL28824030 0.84 DHODH (0.48) KMT2AMEN1HSD11B1ALDH1A1MAPT
SCHEMBL28824037 0.84 MCL1 (0.46) KMT2AMEN1EGLN1HSD11B1ALDH1A1
SCHEMBL29851972 0.82 TSHR (0.44) KMT2AMEN1HSD11B1ALDH1A1MAPT
SCHEMBL28824097 0.82 BCAT2 (0.53) ALDH1A1NPC1HSP90AA1NFKB1RAB9A
SCHEMBL28949290 0.82 DHODH (0.46) MARS1ALDH1A1MAPTL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929676-A Heterocyclic carboxylate compounds as glycolate oxidase inhibitors 紫丁香疗法有限公司 2022-08-19 CN disclosed