SCHEMBL28824030

SCHEMBL28824030

O=C(O)c1cnnn1-c1ccc(-c2ccccc2F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 10/20 0.48
ACMSD Q8TDX5 1/20 0.46
LMNA P02545 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DHFR P00374 1/20 0.40
ALKBH5 Q6P6C2 1/20 0.40
NPC1 O15118 1/20 0.39
HSP90AA1 P07900 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824033 0.86 PTGS1 (0.42) LMNAMAPTNPC1HSP90AA1NFKB1
SCHEMBL28823984 0.85 BRS3 (0.43) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824037 0.84 MCL1 (0.46) ALDH1A1NPC1HSP90AA1NFKB1RAB9A
SCHEMBL28824102 0.84 MAPK9 (0.46) DHODHALDH1A1L3MBTL1NPC1HSP90AA1
SCHEMBL28824043 0.84 KMT2A (0.49) ALDH1A1MAPTL3MBTL1NPC1HSP90AA1
SCHEMBL28824005 0.84 ALDH1A1 (0.42) LMNAALDH1A1NPC1HSP90AA1NFKB1
SCHEMBL29851972 0.82 TSHR (0.44) LMNAALDH1A1MAPTSMN1; SMN2MEN1
SCHEMBL28949290 0.82 DHODH (0.46) DHODHALDH1A1MAPTL3MBTL1NPC1
SCHEMBL28824097 0.82 BCAT2 (0.53) LMNAALDH1A1NPC1HSP90AA1NFKB1
SCHEMBL28824023 0.82 KDM4C (0.44) LMNAALDH1A1MAPTNPC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929676-A Heterocyclic carboxylate compounds as glycolate oxidase inhibitors 紫丁香疗法有限公司 2022-08-19 CN disclosed