SCHEMBL28824079

SCHEMBL28824079

O=C(O)c1cnnn1-c1ccc(-c2ccccc2-c2ncccn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
HSP90AA1 P07900 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD11B1 P28845 6/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
F2 P00734 2/20 0.38
F10 P00742 2/20 0.38
PRSS1 P07477 2/20 0.38
PRSS2 P07478 2/20 0.38
PRSS3 P35030 2/20 0.38
LMNA P02545 2/20 0.37
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824080 0.90 NPC1 (0.40) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824085 0.88 TGFBR1 (0.46) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824102 0.87 MAPK9 (0.46) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28949290 0.85 DHODH (0.46) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824058 0.83 ALOX5AP (0.41) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28823984 0.83 BRS3 (0.43) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824043 0.82 KMT2A (0.49) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824037 0.82 MCL1 (0.46) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824030 0.82 DHODH (0.48) NPC1HSP90AA1NFKB1RAB9ANFKB2
SCHEMBL28824005 0.82 ALDH1A1 (0.42) NPC1HSP90AA1NFKB1RAB9ANFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929676-A Heterocyclic carboxylate compounds as glycolate oxidase inhibitors 紫丁香疗法有限公司 2022-08-19 CN disclosed