SCHEMBL28825528

SCHEMBL28825528

Fc1cccc([CH]c2ccccn2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.53
RAB9A P51151 6/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NFE2L2 Q16236 7/20 0.51
PKM P14618 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPK1 P28482 1/20 0.48
THPO P40225 1/20 0.48
CHRM5 P08912 1/20 0.48
GRM5 P41594 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
ATM Q13315 1/20 0.47
GRM4 Q14833 1/20 0.45
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL711254 0.83 NFE2L2 (0.55) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL711255 0.83 NFE2L2 (0.55) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL28825496 0.79 RAB9A (0.52) NPC1RAB9AMEN1KMT2ANFE2L2
SCHEMBL28825645 0.79 RAB9A (0.47) NPC1RAB9AMEN1KMT2ANFE2L2
SCHEMBL427375 0.78 NPC1 (0.61) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL28825433 0.78 NPC1 (0.42) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL28825486 0.77 NFE2L2 (0.47) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL3300301 0.76 NFE2L2 (0.71) NPC1RAB9ANFE2L2PKMCYP1A2
SCHEMBL28825636 0.75 NFE2L2 (0.55) NPC1RAB9AMEN1KMT2ANFE2L2
SCHEMBL28517481 0.75 PTGS1 (0.50) NPC1RAB9AMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed