SCHEMBL28517481

SCHEMBL28517481

Cc1cc([CH]c2ccccn2)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.50
PTGS2 P35354 1/20 0.50
MEN1 O00255 4/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
KMT2A Q03164 4/20 0.42
ATM Q13315 1/20 0.42
NFE2L2 Q16236 2/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GABRA1 P14867 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
ACHE P22303 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
GRIN1 Q05586 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825645 0.85 RAB9A (0.47) PTGS1PTGS2MEN1NPC1RAB9A
SCHEMBL28516941 0.81 GABRA1 (0.38) PTGS1PTGS2MEN1NPC1RAB9A
SCHEMBL28949583 0.79 GRIN2B (0.36) PTGS1PTGS2NFE2L2GABRA1SIGMAR1
SCHEMBL28825503 0.79 MEN1 (0.41) PTGS1PTGS2MEN1NPC1RAB9A
SCHEMBL28825496 0.75 RAB9A (0.52) MEN1NPC1RAB9AKMT2AATM
SCHEMBL28825467 0.75 GRIN1 (0.42) MEN1NPC1RAB9AKMT2AATM
SCHEMBL28825528 0.75 NPC1 (0.53) PTGS1PTGS2MEN1NPC1RAB9A
SCHEMBL28525691 0.73 ALOX5 (0.44) PTGS1PTGS2MEN1NPC1RAB9A
SCHEMBL27905797 0.72 NPC1 (0.52) MEN1NPC1RAB9AKMT2AATM
SCHEMBL28517024 0.71 ALOX5 (0.50) PTGS1PTGS2NPC1RAB9ANFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026094-B Substituted 4-azaindoles and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2021-02-09 CN claimed
CN-108026094-B Substituted 4-azaindoles and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2021-02-09 CN disclosed