SCHEMBL28825645

SCHEMBL28825645

Fc1ccc([CH]c2ccccn2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.47
MEN1 O00255 3/20 0.47
NPC1 O15118 3/20 0.47
KMT2A Q03164 3/20 0.47
ATM Q13315 1/20 0.47
PLA2G7 Q13093 1/20 0.41
NFE2L2 Q16236 5/20 0.41
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
NR4A1 P22736 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
MAOA P21397 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28517481 0.85 PTGS1 (0.50) RAB9AMEN1NPC1KMT2AATM
SCHEMBL28825503 0.83 MEN1 (0.41) RAB9AMEN1NPC1KMT2AATM
SCHEMBL28825496 0.79 RAB9A (0.52) RAB9AMEN1NPC1KMT2AATM
SCHEMBL28825467 0.79 GRIN1 (0.42) RAB9AMEN1NPC1KMT2AATM
SCHEMBL28825528 0.79 NPC1 (0.53) RAB9AMEN1NPC1KMT2AATM
SCHEMBL28525148 0.77 NFE2L2 (0.40) RAB9AMEN1NPC1KMT2APLA2G7
SCHEMBL27905797 0.76 NPC1 (0.52) RAB9AMEN1NPC1KMT2AATM
SCHEMBL427375 0.74 NPC1 (0.61) RAB9AMEN1NPC1KMT2AATM
SCHEMBL41190 0.73 RAB9A (0.74) RAB9AMEN1NPC1KMT2AATM
SCHEMBL3299908 0.73 NFE2L2 (0.54) RAB9ANPC1KMT2APLA2G7NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed