SCHEMBL711255

SCHEMBL711255

Fc1cccc(C=CC=Cc2ccccn2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 8/20 0.55
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
GRM4 Q14833 1/20 0.50
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ATM Q13315 1/20 0.48
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
PKM P14618 1/20 0.46
MAPK1 P28482 1/20 0.46
THPO P40225 1/20 0.46
CHRM5 P08912 1/20 0.46
GRM5 P41594 1/20 0.46
BLM P54132 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL711254 1.00 NFE2L2 (0.55) NFE2L2NPC1RAB9AMEN1KMT2A
SCHEMBL28825528 0.83 NPC1 (0.53) NFE2L2NPC1RAB9AMEN1KMT2A
SCHEMBL716031 0.81 RAB9A (0.54) NFE2L2NPC1RAB9AMEN1KMT2A
SCHEMBL716032 0.81 RAB9A (0.54) NFE2L2NPC1RAB9AMEN1KMT2A
SCHEMBL709598 0.80 NPC1 (0.48) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL709599 0.80 NPC1 (0.48) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL708639 0.80 NPC1 (0.62) NPC1RAB9AMEN1KMT2AGRM4
SCHEMBL708638 0.80 NPC1 (0.62) NPC1RAB9AMEN1KMT2AGRM4
SCHEMBL715979 0.80 NFE2L2 (0.49) NFE2L2NPC1RAB9AMEN1KMT2A
SCHEMBL715978 0.80 NFE2L2 (0.49) NFE2L2NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124625-B2 enhancing the expression of apoAI; prevention or therapy of dislipidemia SHIONOGI & CO., LTD. (JP) 2012-02-28 US disclosed
US-8053445-B2 Utilities of olefin derivatives SHIONOGI & CO., LTD. (JP) 2011-11-08 US disclosed
US-20090036457-A1 Utilities of olefin derivatives YAMAMORI TERUO 2009-02-05 US disclosed
US-20040242615-A1 Utilities of olefin derivatives SHIONOGI & CO., LTD. (JP) 2004-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040242615-A1 Utilities of olefin derivatives APOL1, NR1H2, APOB NFE2L2 576/4885NPC1 19/4885RAB9A 4723/4885
US-20090036457-A1 Utilities of olefin derivatives APOL1, APOB, NR1H2 NFE2L2 1105/4885NPC1 48/4885RAB9A 4606/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.