SCHEMBL28825629

SCHEMBL28825629

COS(=O)(=O)Cc1ccc(C(F)(F)F)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.41
TRPV4 Q9HBA0 1/20 0.41
KCNH2 Q12809 3/20 0.37
NAMPT P43490 1/20 0.37
PPARD Q03181 1/20 0.37
MAP4K4 O95819 1/20 0.37
PIK3CA P42336 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
TKT P29401 1/20 0.37
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNQ4 P56696 1/20 0.37
KCNQ5 Q9NR82 1/20 0.37
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
PTPRZ1 P23471 1/20 0.36
CYP2C9 P11712 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12797513 0.79 DAO (0.42) DAOTRPV4KCNH2NAMPTMAP4K4
SCHEMBL13373481 0.79 DAO (0.45) DAOTRPV4KCNH2NAMPTMAP4K4
SCHEMBL17979483 0.79 KIF11 (0.51) DAOTRPV4KCNH2NAMPTMAP4K4
SCHEMBL10296101 0.79 TRPV4 (0.44) DAOTRPV4KCNH2NAMPTPPARD
SCHEMBL29271395 0.79 NFE2L2 (0.40) KCNH2
SCHEMBL20508396 0.79
SCHEMBL24425812 0.78 DAO (0.41) DAOTRPV4KCNH2NAMPTMAP4K4
SCHEMBL12464348 0.77 DAO (0.40) DAOTRPV4KCNH2NAMPTMAP4K4
SCHEMBL23141526 0.77 LOXL2 (0.53) KCNQ2
SCHEMBL18571250 0.77 DAO (0.40) DAOTRPV4KCNH2NAMPTMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed