SCHEMBL28825697

SCHEMBL28825697

Fc1cc(F)cc([CH]c2ccc(F)c(C(F)F)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.35
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28686608 0.81 GRIN2B (0.37) NFE2L2GRIN1GRIN2B
SCHEMBL28825574 0.77 GRIN1 (0.37) GRIN1GRIN2B
SCHEMBL28825619 0.75 GRIN2B (0.37) NFE2L2GRIN1GRIN2B
SCHEMBL21020970 0.74 ALDH1A1 (0.42) NFE2L2
SCHEMBL5251881 0.73 PTGS1 (0.42) NFE2L2BACE1
SCHEMBL28825635 0.73 KCNH2 (0.41) GRIN1GRIN2B
SCHEMBL28825504 0.73 ALOX5 (0.42) NFE2L2GRIN1GRIN2B
SCHEMBL28825624 0.72 GRIN2B (0.39) NFE2L2GRIN1GRIN2B
SCHEMBL16954998 0.69 CES2 (0.48) NFE2L2GRIN1GRIN2B
SCHEMBL28825503 0.69 MEN1 (0.41) NFE2L2GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed