SCHEMBL28828362

SCHEMBL28828362

COc1cccc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)c1F

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.40
APP P05067 2/20 0.40
ERN1 O75460 1/20 0.39
FFAR2 O15552 1/20 0.38
CTSA P10619 2/20 0.38
DYRK1A Q13627 1/20 0.37
DHODH Q02127 2/20 0.37
CTSD P07339 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
FAAH O00519 1/20 0.36
PIN1 Q13526 1/20 0.36
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828483 0.91 EDNRB (0.42) BACE1FFAR2CTSDEDNRBEDNRA
SCHEMBL28828528 0.88 ADORA3 (0.38) BACE1CTSAEDNRBEDNRA
SCHEMBL28828386 0.88 CTSA (0.38) CTSADHODHPIN1
SCHEMBL28828489 0.88 PGR (0.38) BACE1APPDYRK1AHDAC6HDAC1
SCHEMBL28828616 0.88 PIN1 (0.43) BACE1APPERN1CTSAPIN1
SCHEMBL28828447 0.88 HSD17B3 (0.37) FFAR2DHODHEDNRBEDNRA
SCHEMBL28950181 0.87 CTSA (0.33) BACE1APPCTSAEDNRBEDNRA
SCHEMBL28828572 0.86 ITGB1 (0.34) CTSA
SCHEMBL28828652 0.85 CTSA (0.37) CTSA
SCHEMBL28828631 0.85 ACMSD (0.37) DYRK1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed