SCHEMBL28828652

SCHEMBL28828652

COc1cc(F)c(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 2/20 0.37
AR P10275 1/20 0.35
KDM1A O60341 2/20 0.34
KDM1B Q8NB78 2/20 0.34
TDP2 O95551 1/20 0.34
PTGS2 P35354 5/20 0.34
PTGS1 P23219 2/20 0.34
FPR2 P25090 1/20 0.33
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
RORC P51449 1/20 0.32
PRKCZ Q05513 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
F2R P25116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828429 0.90 KDM1A (0.33) KDM1AKDM1BPTGS2RORC
SCHEMBL29121288 0.88 TDP2 (0.43) ARTDP2PTGS2PTGS1ABHD6
SCHEMBL28828529 0.88 PDE4A (0.35) KDM1ATDP2F2R
SCHEMBL29121280 0.88 AR (0.42) ARTDP2PTGS2PTGS1PRKCZ
SCHEMBL28828386 0.86 CTSA (0.38) CTSAKDM1A
SCHEMBL28828414 0.86 PTGS2 (0.39) ARPTGS2FPR2PRKAB2PRKAG1
SCHEMBL28828754 0.85 AKR1C3 (0.38) CTSAKDM1AKDM1B
SCHEMBL28828616 0.85 PIN1 (0.43) CTSAFFAR4
SCHEMBL28828390 0.85 FFAR1 (0.42) KDM1AKDM1B
SCHEMBL28828483 0.85 EDNRB (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed