SCHEMBL28828519

SCHEMBL28828519

COc1ccc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)cc1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
S1PR1 P21453 5/20 0.35
RXRA P19793 2/20 0.34
RXRB P28702 2/20 0.34
RXRG P48443 2/20 0.34
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
SLC9A1 P19634 1/20 0.33
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
SLC2A1 P11166 1/20 0.33
ABHD6 Q9BV23 1/20 0.33
F2R P25116 1/20 0.33
PPIB P23284 1/20 0.32
PPIA P62937 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828413 0.89 RXRA (0.48) S1PR1RXRARXRBRXRGCTSS
SCHEMBL29121288 0.86 TDP2 (0.43) ABHD6
SCHEMBL28950193 0.85 PIK3CD (0.41) ITGB2ICAM1ITGALSLC9A1F2R
SCHEMBL28828416 0.85 PTGDR2 (0.40)
SCHEMBL28828534 0.84 PTGS2 (0.39) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL29121269 0.84 PTGS2 (0.39) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28828529 0.84 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DF2R
SCHEMBL28828662 0.84 KIF11 (0.43) SLC9A1
SCHEMBL28828674 0.83 PDE4B (0.35) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28828572 0.81 ITGB1 (0.34) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed