SCHEMBL28828529

SCHEMBL28828529

COc1cc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 4/20 0.35
PDE4B Q07343 4/20 0.35
PDE4C Q08493 4/20 0.35
PDE4D Q08499 4/20 0.35
KDM1A O60341 2/20 0.35
TDP2 O95551 1/20 0.34
F2R P25116 1/20 0.34
GRM4 Q14833 1/20 0.33
MAOA P21397 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
GRK6 P43250 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29121288 0.91 TDP2 (0.43) TDP2CYP3A4
SCHEMBL28828604 0.89 CYP17A1 (0.33) F2RCYP3A4
SCHEMBL28828652 0.88 CTSA (0.37) KDM1ATDP2F2R
SCHEMBL28828674 0.88 PDE4B (0.35) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL28828522 0.87 DYRK1A (0.38) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL28828388 0.86 DAPK3 (0.38) F2R
SCHEMBL28828677 0.86 IKBKB (0.33) F2R
SCHEMBL28828601 0.85 TDP2 (0.39) TDP2
SCHEMBL28828426 0.85 KDM1A (0.39) KDM1AF2RCYP3A4
SCHEMBL28828534 0.84 PTGS2 (0.39) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed