SCHEMBL28828522

SCHEMBL28828522

COc1cc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.38
RIPK2 O43353 1/20 0.37
KMO O15229 1/20 0.37
CHEK1 O14757 1/20 0.36
PDE4A P27815 6/20 0.35
PDE4B Q07343 6/20 0.35
PDE4C Q08493 6/20 0.35
PDE4D Q08499 6/20 0.35
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
FFAR2 O15552 1/20 0.33
GRM4 Q14833 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
MIF P14174 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828534 0.91 PTGS2 (0.39) KMOPDE4APDE4BPDE4CPDE4D
SCHEMBL29121269 0.91 PTGS2 (0.39) KMOPDE4APDE4BPDE4CPDE4D
SCHEMBL29228314 0.89 DYRK1A (0.37) DYRK1ARIPK2KMOCHEK1PDE4A
SCHEMBL28828703 0.89 PGR (0.38) SLC9A1
SCHEMBL29121238 0.88 MKNK1 (0.34) KMOSLC9A1
SCHEMBL28828674 0.88 PDE4B (0.35) KMOPDE4APDE4BPDE4CPDE4D
SCHEMBL28828529 0.87 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL28828686 0.85 SIRT1 (0.36) KMOSLC9A1
SCHEMBL28828640 0.85 SIRT2 (0.36) SLC9A1KDM4EMAPT
SCHEMBL28828363 0.84 CHRNB2 (0.39) TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed