SCHEMBL28828838

SCHEMBL28828838

O=C(Cn1c(-c2ccc(Cl)cc2)c(Cl)[nH]c1=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.40
GRIN2B Q13224 8/20 0.40
AVPR2 P30518 2/20 0.37
AVPR1A P37288 2/20 0.37
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
LMNA P02545 2/20 0.33
HTT P42858 1/20 0.33
MAPT P10636 1/20 0.33
BRD4 O60885 1/20 0.33
BRD2 P25440 1/20 0.33
BRD3 Q15059 1/20 0.33
BRDT Q58F21 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA9 Q16790 1/20 0.32
XBP1 P17861 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28829055 0.87 GRIN1 (0.38) GRIN1GRIN2BAVPR2AVPR1AHDAC2
SCHEMBL28828864 0.87 GRIN1 (0.41) GRIN1GRIN2BAVPR2AVPR1AMAPT
SCHEMBL28828984 0.83 APEX1 (0.46) GRIN1GRIN2B
SCHEMBL28828770 0.77 AVPR2 (0.42) AVPR2AVPR1A
SCHEMBL28828769 0.77 AVPR2 (0.42) AVPR2AVPR1A
SCHEMBL28829027 0.77 ALDH1A1 (0.42) GRIN1GRIN2BAVPR2AVPR1AHDAC2
SCHEMBL28828908 0.76 TSHR (0.50) LMNAHTTMAPT
SCHEMBL168320 0.76 APOBEC3G (0.45) GRIN1GRIN2BAVPR2AVPR1AHDAC2
SCHEMBL28828841 0.69 AKR1B10 (0.44) GRIN1GRIN2B
SCHEMBL28828872 0.69 POLB (0.44) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835688-A Substituted 4-aryl imidazole-2-ketone derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-08-02 CN disclosed