SCHEMBL28828864

SCHEMBL28828864

Cc1[nH]c(=O)n(CC(=O)C(F)(F)F)c1-c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.41
GRIN2B Q13224 8/20 0.41
AVPR2 P30518 2/20 0.40
AVPR1A P37288 2/20 0.40
MAPT P10636 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GRM5 P41594 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828838 0.87 GRIN1 (0.40) GRIN1GRIN2BAVPR2AVPR1AMAPT
SCHEMBL28829055 0.85 GRIN1 (0.38) GRIN1GRIN2BAVPR2AVPR1AMAPT
SCHEMBL28828841 0.84 AKR1B10 (0.44) GRIN1GRIN2B
SCHEMBL28828790 0.80 TSHR (0.50) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL28828912 0.79 AVPR2 (0.43) AVPR2AVPR1A
SCHEMBL28828920 0.79 AVPR2 (0.43) AVPR2AVPR1A
SCHEMBL168320 0.76 APOBEC3G (0.45) GRIN1GRIN2BAVPR2AVPR1AMAPT
SCHEMBL28829027 0.75 ALDH1A1 (0.42) GRIN1GRIN2BAVPR2AVPR1AMAPT
SCHEMBL28828984 0.70 APEX1 (0.46) GRIN1GRIN2BKDM4EALDH1A1HPGD
SCHEMBL28828908 0.69 TSHR (0.50) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835688-A Substituted 4-aryl imidazole-2-ketone derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-08-02 CN disclosed