SCHEMBL28834819

SCHEMBL28834819

COC(=O)c1cc2c(ccn2C2CCOCC2)cc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 5/20 0.44
CFTR P13569 3/20 0.39
DGAT1 O75907 1/20 0.39
GAA P10253 4/20 0.38
HSD17B10 Q99714 4/20 0.38
MAPT P10636 3/20 0.38
HPGD P15428 3/20 0.38
GLA P06280 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
ATM Q13315 1/20 0.38
ABL1 P00519 1/20 0.37
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28834792 0.83 SIRT6 (0.42) ALDH1A1GAAMAPTHPGDLMNA
SCHEMBL27186173 0.78 ALDH1A1 (0.45) ALDH1A1KDM4ECFTRGAAHSD17B10
SCHEMBL28834838 0.77 CNR2 (0.41) ALDH1A1KDM4ECFTRGAAHSD17B10
SCHEMBL29901725 0.77 KDM4E (0.39) ALDH1A1KDM4ECFTRGAAHSD17B10
SCHEMBL15998985 0.75 HTR3A (0.43) ALDH1A1MAPTOPRK1CNR1CNR2
SCHEMBL31438003 0.75 FGFR1 (0.43) ALDH1A1KDM4EGAAHSD17B10MAPT
SCHEMBL21231982 0.74 KDM4E (0.49) ALDH1A1KDM4ECFTRGAAHSD17B10
SCHEMBL20606472 0.74 IRAK4 (0.58) ALDH1A1KDM4EIRAK4
SCHEMBL23530107 0.71 KDM4C (0.37) ALDH1A1KDM4EDGAT1KDM4CIRAK4
SCHEMBL29550517 0.71 KDM4C (0.37) ALDH1A1KDM4EDGAT1KDM4CIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028644-A SOS1 inhibitor heterocyclic compounds 首药控股(北京)股份有限公司 2022-09-09 CN disclosed