SCHEMBL28835206

SCHEMBL28835206

CC(C)(C)C(=O)ON1CCC(Nc2ccc(C#N)cc2N)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.44
IRAK4 Q9NWZ3 3/20 0.39
ALOX15 P16050 2/20 0.39
JAK2 O60674 6/20 0.38
JAK3 P52333 6/20 0.38
JAK1 P23458 5/20 0.38
KCNH2 Q12809 4/20 0.38
SSTR4 P31391 1/20 0.38
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
CLK1 P49759 1/20 0.37
CLK2 P49760 1/20 0.37
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37
IRAK1 P51617 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
DRD2 P14416 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28104989 0.91 GPR119 (0.42) GPR119IRAK4JAK2JAK3JAK1
SCHEMBL27741408 0.84 ALOX15 (0.44) IRAK4ALOX15NOS1NOS2ALDH1A1
SCHEMBL4438915 0.84 GPR119 (0.61) GPR119IRAK4ALDH1A1
SCHEMBL28772407 0.81 ALOX15 (0.42) ALOX15ALDH1A1GAA
SCHEMBL28331009 0.81 GPR119 (0.37) GPR119IRAK4ALOX15JAK2JAK3
SCHEMBL27909355 0.80 MAPT (0.49) ALOX15KDM4EALDH1A1GAA
SCHEMBL7178322 0.80 GPR119 (0.54) GPR119IRAK4ALDH1A1
SCHEMBL7189717 0.80 GPR119 (0.54) GPR119IRAK4ALDH1A1
SCHEMBL7178327 0.80 GPR119 (0.54) GPR119IRAK4ALDH1A1
SCHEMBL7182896 0.79 DRD2 (0.52) GPR119IRAK4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061969-B TRPA1 regulator ALGOMEDIX, INC. (US) 2019-10-29 CN disclosed
CN-106061969-A TRPA1 modulators 阿尔戈么迪克斯有限公司 2016-10-26 CN disclosed