SCHEMBL28836147

SCHEMBL28836147

Cc1cc(N2CCCCC2)nnc1C(=O)NC1CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.60
HSD11B1 P28845 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.48
TAS1R3 Q7RTX0 2/20 0.48
TAS1R1 Q7RTX1 2/20 0.48
TAS1R2 Q8TE23 2/20 0.48
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111732 0.76 CNR2 (0.78) CNR2HSD11B1SMN1; SMN2LMNATSHR
SCHEMBL28111774 0.75 HSD11B1 (0.66) CNR2HSD11B1SMN1; SMN2MEN1CYP1A2
SCHEMBL2591980 0.68 HSD11B1 (1.00) CNR2HSD11B1SMN1; SMN2MEN1CYP1A2
SCHEMBL28836519 0.68 CNR2 (0.53) CNR2LMNATSHRMEN1CYP1A2
SCHEMBL22565386 0.67 ACKR3 (0.61) CNR2HSD11B1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL22449359 0.66 ALDH1A1 (0.64) HSD11B1SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL1014776 0.66 POLB (0.64) HSD11B1SMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL1017870 0.66 POLB (0.64) HSD11B1SMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL12590352 0.66 POLB (0.66) CNR2SMN1; SMN2TSHRCYP1A2CYP3A4
SCHEMBL704712 0.65 TAS1R3 (1.00) SMN1; SMN2TAS1R3TAS1R1TAS1R2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN claimed
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN disclosed