SCHEMBL28840392

SCHEMBL28840392

Cc1nc(OCC(F)(F)F)c(F)cc1CNC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PKM P14618 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SGK1 O00141 1/20 0.32
ALDH1A1 P00352 4/20 0.32
MAPT P10636 1/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
KDM4E B2RXH2 3/20 0.32
HPGD P15428 2/20 0.32
HIF1A Q16665 1/20 0.32
GAA P10253 1/20 0.32
ALOX15 P16050 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27931782 0.84 KCNH2 (0.35) CNR2MAPTDGAT1
SCHEMBL27931827 0.83 CNR2 (0.34) CNR2ACACB
Pyrazinamide SCHEMBL28093474 0.82 ADORA3 (0.40) CNR2KMT2ACYP1A2KDM4EDGAT1
SCHEMBL2714834 0.81 ALDH1A1 (0.34) CNR2MEN1KMT2AALDH1A1MAPT
SCHEMBL2717106 0.81 PTGS2 (0.35) CNR2MEN1KMT2ACYP2C9CYP2C19
SCHEMBL28130155 0.75 MEN1 (0.36) CNR2MEN1KMT2ACYP1A2CYP2C19
SCHEMBL27913875 0.75 KCNH2 (0.47) KMT2AMAPTGAA
SCHEMBL27914078 0.75 MMP13 (0.42) CNR2MEN1KMT2AACACB
SCHEMBL27931958 0.74 CYP1A2 (0.36) CNR2MEN1KMT2ACYP1A2CYP2C9
SCHEMBL18258951 0.73 ACACB (0.36) CNR2MEN1KMT2AMAPTACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478497-A Aryl amine derivatives as TTX S blocker 拉夸里亚创药株式会社 2017-03-08 CN disclosed