SCHEMBL28845665

SCHEMBL28845665

O=C(NCCc1ccccc1)c1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.51
CDK8 P49336 1/20 0.51
GPR52 Q9Y2T5 3/20 0.51
DNMT1 P26358 1/20 0.50
DNMT3A Q9Y6K1 1/20 0.50
KDM5B Q9UGL1 2/20 0.48
KDM4E B2RXH2 1/20 0.48
KDM5A P29375 1/20 0.48
KDM5C P41229 1/20 0.48
NAMPT P43490 1/20 0.45
MLYCD O95822 1/20 0.45
AURKA O14965 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845651 0.89 GPR52 (0.54) GPR52DNMT1DNMT3AGAKALDH1A1
SCHEMBL28845687 0.88 ALDH1A1 (0.57) GPR52DNMT1DNMT3AAURKAGAK
SCHEMBL28845643 0.87 GPR52 (0.59) GPR52DNMT1DNMT3AGAKALDH1A1
SCHEMBL28845637 0.86 DNMT1 (0.52) GPR52DNMT1DNMT3AAURKAGAK
SCHEMBL28845675 0.86 DNMT1 (0.68) DNMT1DNMT3AAURKALMNAGAK
SCHEMBL29140025 0.83 GAK (0.54) GPR52DNMT1DNMT3ALMNAGAK
SCHEMBL28845682 0.82 DNMT1 (0.54) CCNCCDK8DNMT1DNMT3AMLYCD
SCHEMBL29200469 0.80 GAK (0.55) DNMT1DNMT3AAURKAGAKPRKD3
SCHEMBL28845648 0.80 NPSR1 (0.56) GPR52DNMT1DNMT3AAURKAGAK
SCHEMBL28845680 0.79 GAK (0.51) GPR52DNMT1DNMT3AAURKAHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN claimed
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed