SCHEMBL28845802

SCHEMBL28845802

Cc1cc(-c2ccccc2C(N)=O)c(C)c([N+](=O)[O-])c1C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.41
POLB P06746 3/20 0.39
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MAPT P10636 3/20 0.39
TSHR P16473 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.37
CDC7 O00311 1/20 0.37
KDM4E B2RXH2 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BRD4 O60885 1/20 0.36
MYC P01106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27583224 0.81 BCAT2 (0.50) BCAT2ALDH1A1NPC1RAB9AMAPT
SCHEMBL6205026 0.79 TDP1 (0.44) POLBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL29950282 0.72 LMNA (0.54) BCAT2ALDH1A1MAPTTSHRTDP1
SCHEMBL4332774 0.72 ALDH1A1 (0.40) POLBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL30986109 0.72 ALDH1A1 (0.62) POLBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL2636763 0.72 ALDH1A1 (0.62) POLBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL995083 0.72 LMNA (0.54) BCAT2ALDH1A1MAPTTSHRTDP1
SCHEMBL27505005 0.72 TDP1 (0.44) POLBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL17157028 0.72 ALDH1A1 (0.52) BCAT2POLBALDH1A1SMN1; SMN2NPC1
SCHEMBL1788703 0.71 BCAT2 (0.59) BCAT2ALDH1A1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed