SCHEMBL28869814

SCHEMBL28869814

COC(=O)Cc1ccc(NC(=O)Cc2ccc3ccccc3c2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.73
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
L3MBTL1 Q9Y468 2/20 0.62
NLRP3 Q96P20 1/20 0.60
SMN1; SMN2 Q16637 3/20 0.58
ALDH1A1 P00352 2/20 0.58
MAPT P10636 2/20 0.58
RAB9A P51151 2/20 0.58
HPGD P15428 2/20 0.56
LMNA P02545 2/20 0.56
MAPK10 P53779 2/20 0.56
GSK3A P49840 1/20 0.56
RIOK2 Q9BVS4 1/20 0.56
MAPK8 P45983 1/20 0.55
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28869818 0.90 KMT2A (0.75) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL14344626 0.88 MEN1 (0.76) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL31170867 0.87 MEN1 (0.57) NR1H4MEN1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL2662328 0.87 MEN1 (0.57) NR1H4MEN1KMT2AL3MBTL1SMN1; SMN2
Hydrochloric Acid SCHEMBL5846666 0.85 MEN1 (0.56) NR1H4MEN1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL28869822 0.85 RAB9A (0.71) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL13451637 0.85 NR1H4 (0.74) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL13451638 0.85 NR1H4 (0.74) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL28869815 0.85 NR1H4 (0.79) NR1H4MEN1KMT2AL3MBTL1NLRP3
SCHEMBL9367263 0.84 NR1H4 (0.83) NR1H4MEN1KMT2AL3MBTL1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478070-A Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN disclosed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN disclosed