SCHEMBL28869818

SCHEMBL28869818

COC(=O)Cc1cccc(NC(=O)Cc2ccc3ccccc3c2)c1

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.75
MEN1 O00255 3/20 0.75
L3MBTL1 Q9Y468 1/20 0.70
NLRP3 Q96P20 2/20 0.68
USP2 O75604 1/20 0.59
NR1H4 Q96RI1 1/20 0.59
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
HTT P42858 1/20 0.56
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
MAPK10 P53779 2/20 0.54
GSK3A P49840 1/20 0.54
RIOK2 Q9BVS4 1/20 0.54
POLB P06746 1/20 0.53
MAPK8 P45983 1/20 0.53
ANO1 Q5XXA6 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28869814 0.90 NR1H4 (0.73) KMT2AMEN1L3MBTL1NLRP3NR1H4
SCHEMBL28869800 0.85 NLRP3 (0.73) KMT2AMEN1L3MBTL1NLRP3USP2
SCHEMBL31170867 0.85 MEN1 (0.57) KMT2AMEN1L3MBTL1NR1H4SMN1; SMN2
SCHEMBL2662328 0.85 MEN1 (0.57) KMT2AMEN1L3MBTL1NR1H4SMN1; SMN2
SCHEMBL7435795 0.84 NR1H4 (0.64) KMT2AMEN1L3MBTL1NR1H4SMN1; SMN2
SCHEMBL28957115 0.84 MEN1 (0.73) KMT2AMEN1L3MBTL1NLRP3USP2
Hydrochloric Acid SCHEMBL5846666 0.83 MEN1 (0.56) KMT2AMEN1L3MBTL1NR1H4SMN1; SMN2
SCHEMBL9367263 0.82 NR1H4 (0.83) KMT2AMEN1L3MBTL1NLRP3NR1H4
Cyclopropane SCHEMBL11849208 0.81 MEN1 (0.53) KMT2AMEN1L3MBTL1NR1H4SMN1; SMN2
SCHEMBL2038480 0.80 L3MBTL1 (0.76) KMT2AMEN1L3MBTL1NLRP3NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478070-A Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN disclosed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN disclosed