SCHEMBL28871017

SCHEMBL28871017

Brc1ccc(Br)cc1.O=[N+]([O-])c1cc(F)c(F)cc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.50
ATM Q13315 1/20 0.50
ALDH1A1 P00352 4/20 0.48
HIF1A Q16665 1/20 0.48
VCAM1 P19320 1/20 0.46
MAPT P10636 5/20 0.45
PKM P14618 2/20 0.45
MAPK1 P28482 2/20 0.44
S100A4 P26447 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
CYP3A4 P08684 2/20 0.42
TSHR P16473 1/20 0.42
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CASP6 P55212 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30257990 0.86 TDP1 (0.56) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL3756498 0.86 TDP1 (0.56) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL29399835 0.81 TDP1 (0.64) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL40706 0.81 ALDH1A1 (0.62) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL6619 0.81 TDP1 (0.64) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL29429960 0.81 ALDH1A1 (0.62) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL29495221 0.80 MAPT (0.59) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL2536509 0.80 MAPT (0.59) TDP1ATMALDH1A1HIF1AVCAM1
Ethylene SCHEMBL27608389 0.78 TDP1 (0.60) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL1561802 0.77 TSHR (0.56) TDP1ATMALDH1A1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683601-A Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2021-11-23 CN claimed
CN-113683601-B Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2022-09-20 CN disclosed
CN-113683601-A Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2021-11-23 CN disclosed