SCHEMBL28877320

SCHEMBL28877320

C=C(CCc1ccccc1)C(F)(F)Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.47
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
ALDH1A1 P00352 1/20 0.44
FFAR1 O14842 1/20 0.44
CES1 P23141 5/20 0.43
FAAH O00519 3/20 0.43
TDP1 Q9NUW8 3/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC1 Q13547 2/20 0.39
HDAC3 O15379 1/20 0.39
MAPK1 P28482 1/20 0.39
ADRA1A P35348 1/20 0.39
HDAC4 P56524 1/20 0.39
SLC6A3 Q01959 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC10 Q969S8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20973256 0.86 CES1 (0.49) KEAP1POLBGAAALDH1A1FFAR1
SCHEMBL27616806 0.78 ALDH1A1 (0.50) KEAP1POLBALDH1A1FFAR1TDP1
SCHEMBL12195215 0.74 KEAP1 (0.54) KEAP1ALDH1A1FFAR1TDP1HDAC2
SCHEMBL13082819 0.73 KEAP1 (0.58) KEAP1ALDH1A1FFAR1TDP1HDAC2
SCHEMBL7269710 0.73 KEAP1 (0.58) KEAP1ALDH1A1FFAR1TDP1HDAC2
SCHEMBL6067580 0.72 ALDH1A1 (0.53) KEAP1POLBGAAALDH1A1FFAR1
SCHEMBL26028772 0.72 FFAR1 (0.44) KEAP1POLBGAAALDH1A1FFAR1
SCHEMBL16795814 0.71 TDP1 (0.50) KEAP1ALDH1A1FFAR1TDP1HDAC2
SCHEMBL7808017 0.71 KEAP1 (0.55) KEAP1POLBGAAALDH1A1FFAR1
SCHEMBL23406423 0.70 KEAP1 (0.54) KEAP1ALDH1A1FFAR1TDP1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118684548-A Method for selective gem-difluoroallylation of (hetero) aryl phenols or polypeptides 中国科学院上海有机化学研究所 2024-09-24 CN disclosed
CN-115260069-B 3, 3-difluoroallylium salt compound and preparation method and application thereof 中国科学院上海有机化学研究所 2023-10-27 CN disclosed
CN-115260069-A 3,3-difluoroallylonium salt compound and preparation method and application thereof 中国科学院上海有机化学研究所 2022-11-01 CN disclosed