SCHEMBL28878201

SCHEMBL28878201

O=S(=O)(Nc1cc(Cl)ccc1O)c1ccc2ccccc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 3/20 0.64
HSD17B2 P37059 1/20 0.60
MEN1 O00255 7/20 0.60
KMT2A Q03164 7/20 0.60
ALDH1A1 P00352 4/20 0.60
MAPT P10636 3/20 0.60
LMNA P02545 2/20 0.60
GAA P10253 2/20 0.60
TP53 P04637 1/20 0.60
HTT P42858 1/20 0.60
HSD17B10 Q99714 1/20 0.60
PKM P14618 1/20 0.57
ERBB2 P04626 1/20 0.56
HSP90AA1 P07900 1/20 0.56
HSP90AB1 P08238 1/20 0.56
TDP1 Q9NUW8 2/20 0.55
POLB P06746 1/20 0.55
THRB P10828 1/20 0.55
FBP1 P09467 1/20 0.54
HKDC1 Q2TB90 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802646 0.84 ERBB2 (0.77) WDR5HSD17B2MEN1KMT2AALDH1A1
SCHEMBL3260752 0.84 MEN1 (0.62) HSD17B2MEN1KMT2AALDH1A1MAPT
SCHEMBL9942107 0.83 HSD17B2 (0.61) HSD17B2MEN1KMT2AALDH1A1MAPT
SCHEMBL28326526 0.83 MEN1 (0.56) MEN1KMT2AALDH1A1GAAHTT
SCHEMBL9927441 0.83 FBP1 (0.56) MEN1KMT2AALDH1A1PKMERBB2
SCHEMBL9775395 0.82 WDR5 (0.68) WDR5HSD17B2MEN1KMT2AALDH1A1
SCHEMBL14434211 0.79 WDR5 (0.61) WDR5HSD17B2MEN1KMT2AALDH1A1
SCHEMBL3260612 0.79 HKDC1 (0.66) MEN1KMT2AALDH1A1MAPTLMNA
SCHEMBL29858930 0.78 WDR5 (1.00) WDR5HSD17B2MEN1KMT2AALDH1A1
SCHEMBL10013441 0.78 MEN1 (0.60) MEN1KMT2AALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110452183-A A kind of preparation method of chiral heterocycle compound SHANGHAI INST ORGANIC CHEMISTRY CAS 2019-11-15 CN disclosed