SCHEMBL28889245

SCHEMBL28889245

COc1cccc(C(C#N)c2cc(C(F)(F)F)ccn2)c1F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.37
ADRB2 P07550 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
AR P10275 3/20 0.34
GAK O14976 1/20 0.34
FYN P06241 1/20 0.33
GAA P10253 1/20 0.33
KRAS P01116 1/20 0.33
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28994023 0.91 KDM4E (0.41) KDM4EMEN1KMT2AATMADRB2
SCHEMBL28889345 0.84 ADRB2 (0.37) KDM4EMEN1KMT2AADRB2ALDH1A1
SCHEMBL28889369 0.81 ADRB2 (0.38) KDM4EMEN1KMT2AATMADRB2
SCHEMBL28889282 0.79 ALDH1A1 (0.40) KDM4EMEN1KMT2AADRB2ALDH1A1
SCHEMBL28889197 0.78 ADRB2 (0.38) KDM4EADRB2ALDH1A1GAA
SCHEMBL28889210 0.78 ADRB2 (0.40) KDM4EMEN1KMT2AADRB2ALDH1A1
SCHEMBL28889190 0.78 ADRB2 (0.40) KDM4EADRB2ALDH1A1ARGAA
SCHEMBL28889153 0.77 ADRB2 (0.40) KDM4EADRB2ALDH1A1GAA
SCHEMBL28889203 0.76 ALDH1A1 (0.50) KDM4EATMADRB2ALDH1A1SMN1; SMN2
SCHEMBL28889348 0.75 GAA (0.42) KDM4EADRB2ALDH1A1GPBAR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed